Quercetin derivatives as novel antihypertensive agents: Synthesis and physiological characterization
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چکیده
منابع مشابه
Quercetin derivatives as novel antihypertensive agents: Synthesis and physiological characterization.
The antihypertensive flavonol quercetin (Q1) is endowed with a cardioprotective effect against myocardial ischemic damage. Q1 inhibits angiotensin converting enzyme activity, improves vascular relaxation, and decreases oxidative stress and gene expression. However, the clinical application of this flavonol is limited by its poor bioavailability and low stability in aqueous medium. In the aim to...
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ژورنال
عنوان ژورنال: European Journal of Pharmaceutical Sciences
سال: 2016
ISSN: 0928-0987
DOI: 10.1016/j.ejps.2015.11.021